1. Theliatinib (HMPL-309) | EGFR 抑制剂 | 现货供应 | 美国品牌Theliatinib (HMPL-309)是一种高效的EGFR抑制剂,对EGFR的Ki值为0.05 nM,对EGFR和EGFR T790M/L858R突变体的IC50值分别为3 nM和22 nM。它对EGFR的选择性是对其他72种激酶的50倍以上。 Quality confirmed by NMR & HPLC. See ...
2. 深入解析——阿法替尼BIBW2992Akihiro Tamiya回顾分析了阿法替尼治疗11例EGFG突变脑膜转NSCLC的情况,绝大多数患者之前均接受过化疗和EGFR-TKI治疗,检测了4例患者的脑脊液EGFR基因突变,均无T790M突变。11例患者中2例肿瘤部分缓解,无进展时间分别为309天和171天,见表3...
3. BIBW2992, an irreversible EGFR/HER2 inhibitor highly...Here, we show that BIBW2992, an anilino-quinazoline designed to irreversibly bind EGFR and HER2, potently suppresses the kinase activity of wild-type and activated EGFR and HER2 mutants, including erlotinib-resistant ...
4. 飞行轨迹 ? C-FIBW 2022年 09月 22日 (KIAH-CYYC) -星期五 05:46:42 51.3288 -113.9351 ← 271° 213 394 2,309 -229 FlightAware ADS-B (CYYC) 星期五 05:46:58 51.3281 -113.9584 ← 260° 208 385 2,256 -229 FlightAware ADS-B 星期五 05:47:14 51.3203 -113.9794...
5. ...support SC - pan_lwip_httpNew issue Link key based on SC, but remote does not support SC - pan_lwip_http_server.c bug #309 Closed naliekkez opened this issue Aug 6, 2020· 12 comments Comments...